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Catalytic hydrogenation in the process of 2-((1-benzylpiperidin-4-yl) methyl)-5,6-dimethoxy-2,3-dihydroinden-1-one hydrochloride synthesis I. Catalyst screening and finding the optimal reaction conditions Cover

Catalytic hydrogenation in the process of 2-((1-benzylpiperidin-4-yl) methyl)-5,6-dimethoxy-2,3-dihydroinden-1-one hydrochloride synthesis I. Catalyst screening and finding the optimal reaction conditions

Open Access
|Oct 2012

References

  1. 1. The American Society of Health- System Pharmacists, AHFS® Consumer Medication Information. ©Copyright, 2010. http://www.ncbi.nlm.nih.gov/pubmedhealth/?term=donepezil.
  2. 2. Gutman, A.L., Shokolnik, E., Tishin, B., Nisnevich, G. & Zaltzman, I. (2002). U.S. Patent No. 6,492,522. Washington, D.C.: U.S. Patent and Trademark Offi ce.
  3. 3. Lerman, O., Kaspi, J., Arad, O., Alnabari, M. & Sery. Y. (2004). U.S. Patent No. 6,844,440. Washington, D.C.: U.S. Patent and Trademark Offi ce.
  4. 4. Reddy, M.S., Eswaraiah, S., Thippannachar, M.V., Chandrashekar, E.R.R., Kumar, P.A.,Kumar, K.N. (2001). U.S. Patent No. 7,148,354. Washington, D.C.: U.S. Patent and Trademark Offi ce.
  5. 5. Iimura, Y. (2001), U.S. Patent No. 6,252,081. Washington, D.C.: U.S. Patent and Trademark Offi ce.
  6. 6. Yatendra, K., Mohan, P., Asok, N. & Nitin, M. WO Patent No. 2004082685(A1). World Intellectual property organization.
  7. 7. Sugimoto, H., Ogura, H., Arai,Y., Limura, Y., Yamanishi, Y. (2002). Research and development of donepezil hydro-chloride, a new type of acetylcholinesterase inhibitor, Jap. J.Pharmacology. 89, 7-20.
  8. 8. Niphade, N., Mali, A., Jagtap, K., Ojha, R.C., Vankawala, P.J. & Mathad, V.T. (2008). Org. Process Res. Dev. 12 (4), 731-735. DOI/10.1021/op800066m.10.1021/op800066m
  9. 9. Attanti, S. & Yadla, V. WO Patent No. /2008/010235. World Intellectual property organization.
  10. 10. Ashvin, K., Aggarwal, C., Vankatesran, S. & Lalit, W. US Patent No. 20100113793, Washington, D.C.: U.S. Patent and Trademark Offi ce.
  11. 11. Thippannachar, M.V., Chintaman, N.N., Jayndal, V.P. & Chaturlal, M.A. Indian Patent Application no. 1073/MUM/2008.
  12. 12. Reichardt, C. (1990). Solvents and Solvent Effects inOrganic Chemistry; VCH: Weinheim,
  13. 13. Rajadhyaksha, R.A. & Karwa, S.L. (1986). Solvents effects in catalytic hydrogenation. Chem.Eng.Sci. 41, 1765. DOI: 10.1016/0009-2509(86)87055-5.10.1016/0009-2509(86)87055-5
  14. 14. McClellan, A.L. (1963). Tables of Experimental DipoleMoments, Vol. I; Freeman and Co., San Francisco, DOI: 10.1002/ange.19650770627.10.1002/ange.19650770627
  15. 15. Singh, U.K. & Vanice, M.A. (2001). Kinetics of liquid-phase hydrogenation reaction over supported metal catalysts. Appl.Catal. A: Gen. 213, 1-24. DOI: 10.1016/S0926-860X(00)00885-1.10.1016/S0926-860X(00)00885-1
  16. 16. Cerveny, L. & Ruzicka, V.; Catal. Rev.-Sci.Eng. 1982, 24, 503-566.
  17. 17. Bakker, J.J.W., Van der Neut, A.G., Kreutzer, M.T., Moulijin, J.A. & Kapteijn, F. (2010). Catalyst performance changes induced by palladium phase transformation in the hydrogenation of benzonitrile. J. Catal. 274, 176-191. DOI: 10.1016/j.cat.2010.06.013.
  18. 18. Bernas, H., Taskinen, A., Wärnå, J. & Murzin, Y. (2009). Hydrogenolysis of hydroxymatairesinol on a Pd/C catalyst. J. Mol. Catal. A: Chem. 306, 33-39, DOI: 10.1016/j. molcata.2009.02.015.
  19. 19. Meitzner, G., Mykyta, W.E.J. & Sinfelt, J.H. (1996). Methylamine hydrogenolysis on a rhodium catalyst-kinetics at high hydrogen partial pressures. Catal. Lett. 37, No.3-4,137-141. DOI: 10.1007/BF00807744. 10.1007/BF00807744
Language: English
Page range: 38 - 47
Published on: Oct 31, 2012
Published by: West Pomeranian University of Technology, Szczecin
In partnership with: Paradigm Publishing Services
Publication frequency: 4 issues per year

© 2012 Zrinka Mastelic Samardzic, Stanka Zrncevic, published by West Pomeranian University of Technology, Szczecin
This work is licensed under the Creative Commons License.