Heterocyclic compounds based on 3-(4-bromophenyl) azo-5-phenyl-2(3H)-furanone: Anti-avian influenza virus (H5N1) activity / Heterociklički derivati 3-(4-bromfenil) azo-5-fenil-2(3H)-furanona: Djelovanje na virus ptičje gripe (H5N1)

Flefel, Eman M.; Abdel-Mageid, Randa E.; Tantawy, Waled A.; Ali, Mohamed A.; Amr, Abd El-Galil E.

doi:10.2478/v10007-012-0037-7

References

1. A. I. Hashem, A. S. A. Youssef, K. A. Kandeel and W. S. I. Abou-Elmaged, Conversion of some 2(3H)-furanones bearing a pyrazolyl group into other heterocyclic systems with a study of their antiviral activity, Eur. J. Med. Chem. 42 (2007) 934-939; DOI: 10.1016/j.ejmech.2006.12.032.10.1016/j.ejmech.2006.12.03217321008
Search in Google Scholar
2. A. I. Hashem, K. A. Kandeel, A. S. A. Youssef and W. S. I. Abou-Elmaged, Behaviour of some 2(3H)-furanones bearing a pyrazolyl group as alkylating agents, J. Chem. Res. 3 (2006) 315-317; DOI: 10.3184/030823406777411115.10.3184/030823406777411115
Search in Google Scholar
3. M. S. Christodoulou, S. Liekens, K. M. Kasiotis and S. A. Haroutounian, Novel pyrazole derivatives: Synthesis and evaluation of anti-angiogenic activity, Bioorg. Med. Chem. 18 (2010) 4338-4350; DOI: 10.1016/j.bmc.2010.04.076.10.1016/j.bmc.2010.04.07620493716
Search in Google Scholar
4. A. Y. Shaw, H. H Liau, P. J. Lu, C. N. Yang, C. H. Lee, J. Y. Chen, Z. Xu and G. Flynn, 3,5-Diaryl-1H-pyrazole as a molecular scaffold for the synthesis of apoptosis-inducing agents, Bioorg. Med. Chem. 18 (2010) 3270-3278; DOI: 10.1016/j.bmc.2010.03.016.10.1016/j.bmc.2010.03.01620381360
Search in Google Scholar
5. J. Choi, Y. Park, H. S. Lee, Y. Yang and S. Yoon, 1,3-Diphenyl-1H-pyrazole derivatives as a new series of potent PPARg partial agonists, Bioorg. Med. Chem. 18 (2010) 8315-8323; DOI: 10.1016/j.bmc.2010.09.068.10.1016/j.bmc.2010.09.06821030263
Search in Google Scholar
6. A. Mohammad, K. Harish and S. A. Javed, Pharmacological activities of pyrazole and its derivatives, Hamdard Medicus 52 (2009) 102-118.
Search in Google Scholar
7. A. El Maatougui, J. Azuaje, E. Sotelo, O. Caamaño and A. Coelho, Silica-supported aluminum chloride-assisted solution phase synthesis of pyridazinone-based antiplatelet agents, ACS Comb. Sci. 10 (2011) 7-12.10.1021/co100017h21247118
Search in Google Scholar
8. A. A. Siddiqui, R. Mishra, M. Shaharyar, A. Husain, M. Rashid and P. Pal, Triazole incorporated pyridazinones as a new class of antihypertensive agents: Design, synthesis and in vivo screening, Bioorg. Med. Chem. Lett. 21 (2011) 1023-1026; DOI: 10.1016/j.bmcl.2010.12.028.10.1016/j.bmcl.2010.12.02821211966
Search in Google Scholar
9. I. H. R. Tomi, A. H. J. Al-Qaisi and Z. H. J. Al-Qaisi, Synthesis, characterization and effect of bis-1,3,4-oxadiazole rings containing glycine moiety on the activity of some transferase enzymes, J. King Saud. Univ. Sci. 23 (2011) 23-33; DOI: 10.1016/j.jksus.2010.06.002.10.1016/j.jksus.2010.06.002
Search in Google Scholar
10. U. Ghani and N. Ullah, New potent inhibitors of tyrosinase: Novel clues to binding of 1,3,4-thiadiazole-2(3H)-thiones, 1,3,4-oxadiazole-2(3H)-thiones, 4-amino-1,2,4-triazole-5(4H)-thiones, and substituted hydrazides to the dicopper active site, Bioorg. Med. Chem. 18 (2010) 4042-4048; DOI: 10.1016/j.bmc.2010.04.021.10.1016/j.bmc.2010.04.02120452224
Search in Google Scholar
11. X. J. Zou, L. H. Lai, G. Y. Jin and Z. X. J. Zhang, Synthesis, fungicidal activity, and 3D-QSAR of pyridazinone-substituted 1,3,4-oxadiazoles and 1,3,4-thiadiazoles, Agr. Food Chem. 50 (2002) 3757-3760; DOI: 10.1021/jf0201677.10.1021/jf020167712059155
Search in Google Scholar
12. G. V. S. Kumar, Y. Rajendraprasad, B. P. Mallikarjuna, S. M. Chandrashekar and C. Kistayya, Synthesis of some novel 2-substituted-5-[isopropylthiazole clubbed] 1,2,4-triazole and 1,3,4-oxadiazoles as potential antimicrobial and antitubercular agents, Eur. J. Med. Chem. 45 (2010) 2063-2074; DOI: 10.1016/j.ejmech.2010.01.045.10.1016/j.ejmech.2010.01.04520149496
Search in Google Scholar
13. K. Imtiaz, A. Sajid, H. Shahid, H. R. Nasim, T. H. Muhammad, W. Abdul, U. Reaz, U. Zaheer, K. Ajmal, A. M. Sajjad and C. Iqbal, Synthesis, antioxidant activities and urease inhibition of some new 1,2,4-triazole and 1,3,4-thiadiazole derivatives, Eur. J. Med. Chem. 45 (2010) 5200-5207; DOI: 10.1016/j.ejmech.2010.08.034.10.1016/j.ejmech.2010.08.03420828889
Search in Google Scholar
14. M. McDowell, S. R. Gonzales, S. C. Kumarapperuma, M. Jeselnik, J. B. Arterburn and K. A. Hanley, A novel nucleoside analog, 1-b-D-ribofuranosyl-3-ethynyl-[1,2,4]triazole (ETAR), exhibits efficacy against a broad range of flaviviruses in vitro, Antivir. Res. 87 (2010) 78-80; DOI: 10.1016/j.antiviral.2010.04.007.10.1016/j.antiviral.2010.04.007289203620416341
Search in Google Scholar
15. H. P. Hsieh and J. T. Hsu, Pyrazole compound BPR1P0034 with potent and selective anti-influenza virus activity, Curr. Pharm. Design 13 (2007) 3531-3542; DOI: 10.1186/1423-0127-17-13.10.1186/1423-0127-17-13283876120178582
Search in Google Scholar
16. A. E. Rashad, A. H. Shamroukh, R. E. Abdel-Megeid, A. Mostafa, M. A. Ali and K. Banert, A facile synthesis and anti-avian influenza virus (H5N1) screening of some novel pyrazolopyrimidine nucleoside derivatives, Nucleos. Nucleot. Nucl. 29 (2010) 809-820; DOI: 10.1080/15257770.2010.529480.10.1080/15257770.2010.52948021128168
Search in Google Scholar
17. K. Hertogs, M. P. Béthune, V. Miller, T. Ivens, P. Schel, A. Van Cauwenberge, C. Van den Eynde, V. van Gerwen, H. Azijn, M. van Houtte, F. Peeters, S. Staszewski, M. Conant, S. Bloor, S. Kemp, B. Larder and R. Pauwels, A rapid method for simultaneous detection of phenotypic resistance to inhibitors of protease and reverse transcriptase in recombinant human immunodeficiency virus type 1 isolates from patients treated with antiretroviral drugs, Antimicrob. Agents Chemother. 42 (1998) 269-276.10.1128/AAC.42.2.2691053999527771
Search in Google Scholar
18. F. G. Hayden, Plaque inhibition assay for drug susceptibility testing of influenza viruses, Agents Chemother. 17 (1980) 865-870.10.1128/AAC.17.5.8652838897396473
Search in Google Scholar

Heterocyclic compounds based on 3-(4-bromophenyl) azo-5-phenyl-2(3H)-furanone: Anti-avian influenza virus (H5N1) activity / Heterociklički derivati 3-(4-bromfenil) azo-5-fenil-2(3H)-furanona: Djelovanje na virus ptičje gripe (H5N1)

References

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