Skip to main content
Have a personal or library account? Click to login
Synthesis and biological evaluation of thieno[2,3-d]pyrimidine derivatives for anti-inflammatory, analgesic and ulcerogenic activity Cover

Synthesis and biological evaluation of thieno[2,3-d]pyrimidine derivatives for anti-inflammatory, analgesic and ulcerogenic activity

Acta Pharmaceutica
Volume 57 (2007): Issue 4 (December 2007)
By: ,   and    
Open Access
|Dec 2007
References

References

  1. D. J. Brown,, in(Ed. A. R. Katritzky and C. W. Rees), Vol., Pergamon Press, Oxford 1984, p. 443.
    Open DOISearch in Google Scholar
  2. B. Roth and C. Cheng,, in(Eds. G. B. Ellis and G. E. West), Vol., Elsevier Biomedical Press, New York 1982, p. 267.
    Search in Google Scholar
  3. M. S. A. E.-A. El-Gaby, S. G. Abdel-Hamide, M. M. Ghorab and S. M. El-Sayed, Synthesis and anticancer activityof some new pyrimidines,(1999) 149-158.
    Search in Google Scholar
  4. C. R. Petrie, H. B. Cottam, P. A. Mckernan, R. K. Robins and G. R. Revankar, Synthesis and biological activity of 6-azacadeguomycin and certain 2,4,6-trisubstituted pyrazolo[3,4-]-pyrimidine ribonucleosides,(1985) 1010-1016.
    Open DOISearch in Google Scholar
  5. M. N. Nasr and M. M. Gineinah, Pyrido[2,3-]pyrimidines and pyrimido[5',4':5,6]-pyrido[2,3-] pyrimidines as new antiviral agents: Synthesis and biological activity,(2002) 289-295; DOI: 10.1002/1521-4184(200208)335:6 289.
    Search in Google Scholar
  6. P. G. Baraldi, M. G. Pavani, M. Nunez, P. Brigidi, B. Vitali, R. Gambari and R. Romagnoli, Antimicrobial and antitumor activity of N-heteroimine-1,2,3-diathiazoles and their transformation in triazolo-, imidazo- and pyrazolopyrimidines,(2002) 449-456; DOI: 10.1016/S0968-0896(01)00294-2.
    Open DOISearch in Google Scholar
  7. S. M. Sondhi, M. Johar, S. Rajvanshi, S. G. Dastidar, R. Shukla, R. Raghubir and J. W. Lown, Anticancer, anti-inflammatory and analgesic activity evaluation of heterocyclic compounds synthesized by the reaction of 4-isothiocyanato-4-methylpentan-2-one with substituted-phenylenediamines,-diaminopyridine and (un)substituted-diamino-pyrimidines,(2001) 69-74; DOI: 10.1071/CH00141.
    Open DOISearch in Google Scholar
  8. A. Z. M. S. Chowdhury, M. M. Matin and M. N. Anwar, Synthesis and antimicrobial activities of fused pyrimidines: Benzothieno[2,3-]imidazol[1,2-c]pyrimidine,(1997) 79-83; ref(1999) 237530p.
    Search in Google Scholar
  9. A. M. Abdel-Fattah, A. S. Aly, F. A. Gad, M. E. A. Zaki and A. B. A. El-Gazzar, A facile synthesis of isooxazolo[5,4:4',5']thiazolo[3,2-]thienopyrimidines, a new ring system,(1998) 263-281; DOI: 10.1080/10426509808033738.
    Open DOISearch in Google Scholar
  10. A. M. Abdel-Fattah, A. S. Aly, F. A. Gad, N. A. Hassan and A. B. A. El-Gazzar, Synthesis and reaction of polynuclear heterocycles, with a new ring system,(2000) 1-27; DOI: 10.1080/10426500008046607.
    Open DOISearch in Google Scholar
  11. A. K. Gewald, E. Schinke and H. Bottcher, 2-Amino-thiophene aus methylenaktiven Nitrilen, Carbonylverbindungen und Schwefel,(1966) 94-100.
    Open DOISearch in Google Scholar
  12. P. Wolkoff, T. S. Nemeth and S. M. Gibson, Reaction of hydrazonyl halides with derivatives of thiourea and thiosemicarbazide; A new source of C-amino- and C-hydrazino-1,2,4-triazoles,(1975) 3211-3215.
    Open DOISearch in Google Scholar
  13. A. F. Hegarty, M. Cashoman, J. B. Aylward and F. L. Scott,-group participation in azocarbonium ion and 1,3-dipolar ion formation,(1971) 1879-1883.
    Open DOISearch in Google Scholar
  14. , Vol., 2ed. (Eds. E. D. Olfert, B. M. Cross and A. A. McWilliam), Canadian Council of Animal Care, Ottawa 1993.
    Search in Google Scholar
  15. C. A. Winter, E. A. Risley and G. W. Nuss, Carrageenin-induced edema in hind paw of the rats as an assay anti-inflammatory drugs,(1962) 544-547.
    Open DOISearch in Google Scholar
  16. J. Miño, V. Moscatelli, O. Hnatyszyn, S. Gorzalczany, C. Acevedo and G. Ferraro, J.(2004) 59-63; DOI: 10.1016/j.phrs.2003.12.016.
    Open DOISearch in Google Scholar
  17. H. D. J. Collier, L. C. Dinnin, C. A. Johnson and C. Schneider., The abdominal response and its suppression by analgestic drugs in the mouse(1968) 295-310.
    Search in Google Scholar
  18. R. K. Goel, A. Chakrabarthi and A. K. Sanyal,(1985) 85-88.
    Open DOISearch in Google Scholar
  19. H. Shay, S. A. Komarav, S. E. Fels, D. Meraza, M. Gruenstein and H. Siplet,(1994) 43-61.
    Search in Google Scholar
  20. A. K. Ganguly and O. P. Bhatnagar,(1973) 748-750.
    Open DOISearch in Google Scholar
  21. A. M. Abdel-Fattah, A. S. Aly, F. Abdel-Motti, N. A. Hassan and H. A. Aly, Synthesis and reaction of some thienopyrimidine derivatives and some of photooxidation,(1995) 627-633.
    Search in Google Scholar
  22. A. S. Aly, A. B. A. El-Gazzar and H. A. R. Hussien, Synthesis and reactions of polynuclear heterocycles: Azolothienopyrimidines and thienothiazolopyrimidines,(2006) 2771-2784; DOI: 10.1080/10426500600865293.
    Open DOISearch in Google Scholar
  23. A. B. A. El-Gazzar, H. A. R. Hussien and A. S. Aly, Synthesis of some derivatives derived from 1,2,3,4-tetrahydrocyclo-hepteno[4,5]thieno[2,3-]pyrimidine,(2007) 35-56; DOI: 10.1080/10426500600864536.
    Open DOISearch in Google Scholar
  24. B. Cacciari and G. Spalluto, Facile and versatile route to the synthesis of fused 2-pyridones: Useful intermediates for polycyclic systems,(2006) 1177-1183; DOI: 10.1080/00397910500514063.
    Open DOISearch in Google Scholar
DOI: https://doi.org/10.2478/v10007-007-0032-6 | Journal eISSN: 1846-9558 | Journal ISSN: 1330-0075
Journal RSS Feed
Language: English, Croatian
Page range: 395 - 411
Published on: Dec 28, 2007
Published by: Croatian Pharmaceutical Society
In partnership with: Paradigm Publishing Services
Keywords:
triazolothienopyrimidine,
thienopyrimidines,
thieno[2,3-d][1,3]thiazine,
thienopyridines,
analgesic,
anti-inflammatory,
ulcerogenic activity
Related subjects:
Pharmacy,
Pharmacy, other

© 2007 Abdel-Rahman El-Gazzar, Hoda Hussein, Hend Hafez, published by Croatian Pharmaceutical Society
This work is licensed under the Creative Commons License.

Volume 57 (2007): Issue 4 (December 2007)
Previous article
Next article