Have a personal or library account? Click to login
Synthesis, antimicrobial and anti-cancer activities of some new N-ethyl, N-benzyl and N-benzoyl-3-indolyl heterocycles Cover

Synthesis, antimicrobial and anti-cancer activities of some new N-ethyl, N-benzyl and N-benzoyl-3-indolyl heterocycles

Open Access
|Jun 2012

References

  1. B. Ngameni, J. Watchueng, F. F. Boyom, F. Keumedjio, B. T. Ngadjui, J. Gut, B. M. Abegaz and P. J. Rosenthal, Antimalarial prenylated chalcones from the twigs of Dorstenia barteri var. subtriangularis, ARKIVOC xiii (2007) 116-123.10.3998/ark.5550190.0008.d14
  2. D. E. Okwu and N. Ukanwa, Isolation and characterization of flavonoids chalcones and anthocynidines from bridelia ferruginea benth, Chem. Sin. 1 (2010) 21-28.
  3. N. Sunduru, A. Agarwal, S. B. Katiyar, Nishi, N. Goyal, S. Gupta and P. M. S. Chauhan, Synthesis of 2,4,6-trisubstituted pyrimidine and triazine heterocycles as antileishmanial agents, Bioorg. Med. Chem. 14 (2006) 7706-7715; DOI: 10.1016/j.bmc.2006.08.009.10.1016/j.bmc.2006.08.00916945542
  4. A. Aitmambetov and Z. Menlimuratova, Interaction of synthetic analogues of natural chalcones and flavones with guanidine, Russ. J. Bioorg. Chem. 29 (2003) 175-176.10.1023/A:1023216600889
  5. M. F. El Shehry, R. H. Swellem, Sh. M. Abu-Bakr and E. M. El-Telbani, Synthesis and molluscicidal evaluation of some new pyrazole, isoxazole, pyridine, pyrimidine, 1,4-thiazine and 1,3,4-thiadiazine derivatives incorporating benzofuran moiety, Eur. J. Med. Chem. 45 (2010) 4783-4787; DOI: 10.1016/j.ejmech.2010.07.043.10.1016/j.ejmech.2010.07.04320801555
  6. A. A. H. Abdel-Rahman, A. E. S. Abdel-Megied, M. A. M. Hawata, E. R. Kasem and M. T. Shaaban, Synthesis and antimicrobial evaluation of some chalcones and their derived pyrazoles, pyrazolines, isoxazolines, and 5,6-dihydropyrimidine-2-(1H)-thiones, Monatsh. Chem. 138 (2007) 889-897; DOI: 10.1007/s00706-007-0700-8.10.1007/s00706-007-0700-8
  7. V. T. Sreevidya, B. Narayana and H. S. Yathirajan, Synthesis and characterization of some chalcones and their cyclohexenone derivatives, Central Eur. J. Chem. 8 (2010) 174-181; DOI: 10.2478/s11532-009-0124-x.10.2478/s11532-009-0124-x
  8. S. George, M. P. Waran, A. Chakraborty and T. K. Ravi, Synthesis and evaluation of the biological activities of some 3-[5-(6-methyl-4-aryl-2-oxo-1,2,3,4-tetrahydropyrimidin-5-yl)-1,3,4-oxadiazol-2-yl]-imino-1,3-di-hydro-2H-indol-2-one derivatives, Acta Pharm. 58 (2008) 119-129; DOI: 10.2478/v10007-007-0050-4.10.2478/v10007-007-0050-418337213
  9. A. H. Mandour, E. R. El-Sawy, K. H. Shaker and M. A. Mustafa, Synthesis, anti-inflammatory, analgesic and anticonvulsant activities of 1,8-dihydro-1-aryl-8-alkyl pyrazolo(3,4-b)indole, Acta Pharm. 60 (2010) 73-88; DOI: 10.2478/v10007-010-0009-8.10.2478/v10007-010-0009-820228042
  10. E. R. El-Sawy, F. A. Bassyouni, S. H. Abu-Bakr, H. M. Rady and M. M. Abdlla, Synthesis and biological activity of some new 1-benzyl and 1-benzoyl 3-heterocyclic indole derivatives, Acta Pharm. 60 (2010) 55-71; DOI: 10.2478/v10007-010-0004-0.10.2478/v10007-010-0004-020228041
  11. A. L. Mndzhoyan, G. L. Papayan, L. D. Zhuruli, S. G. Karagezyan, L. S. Galstyan and V. G. Sarafyan, Synthesis and biological study of hydrazinohydrazones of indole aldehydes and ketones series, Arm. Khim. Zh. (USSR) 22 (1969) 707-713; ref. Chem. Abstr. 72 (1970) 11189f.
  12. A. W. Bauer, W. W. M. Kirby, J. C. Sherris and M. Turck, Antibiotic susceptibility testing by a standardized single disc method, Am. J. Clin. Pathol. 36 (1966) 493-496.10.1093/ajcp/45.4_ts.493
  13. A. H. Moubasher, Soil Fungi in Qatar and other Arab Countries: Aspergillus fumigatus group, Center of Scientific and Applied Research, University of Qatar, Doha 1993, pp. 78-80.
  14. T. Mosmann, Rapid colorimetric assay for cellular growth and survival: application to proliferation and cytotoxicity assays, J. Immunol. Meth. 65 (1983) 55-63; DOI: 10.1038/nbt089.716.
  15. A. Garcia-Raso, J. A. Garcia-Raso, R. Mestres and J. V. Sinisterra, Mechanism of Michael addition of ethyl acetoacetate to chalcone catalyzed by activated Ba(OH)2, React. Kinet. Catal. L. 28 (1985) 365-371; DOI: 10.1007/BF02062966.10.1007/BF02062966
DOI: https://doi.org/10.2478/v10007-012-0020-3 | Journal eISSN: 1846-9558 | Journal ISSN: 1330-0075
Language: English
Page range: 157 - 179
Published on: Jun 28, 2012
Published by: Croatian Pharmaceutical Society
In partnership with: Paradigm Publishing Services
Publication frequency: 4 issues per year
Related subjects:

© 2012 Eslam El-Sawy, Adel Mandour, Khaled Mahmoud, Inas Islam, Heba Abo-Salem, published by Croatian Pharmaceutical Society
This work is licensed under the Creative Commons License.

Volume 62 (2012): Issue 2 (June 2012)