Spherical crystallization of drugs
By: Borut Kovačič, Franc Vrečer and Odon Planinšek
Open Access
|Apr 2012References
- M. K. Franchini,, in(Ed. J. Swarbrick), 3rd ed., Taylor & Francis, New York 2006, DOI: 10.1081/E-EPT-120030638.
- J. C. Chaumeil, Micronization: A method of improving the bioavailability of poorly soluble drugs,(1998) 211-215.
- J. C. Feeley, P. York, B. S. Sumby and H. Dicks, Determination of surface properties and flow characteristics of salbutamol sulphate, before and after micronization,(1998) 89-96; DOI: 10.1016/S0378-5173(98)00179-3.
- M. M. de Villiers, Influence of cohesive properties of micronized drug powders on particle size analysis,(1995) 191-198; DOI: 10.1016/0731-7085(95)01274-O.
- A. K. Tiwary,, in(Ed. J. Swarbrick), 3rd ed., Taylor & Francis, New York 2006, pp. 820-833; DOI: 10.1081/E-EPT-120019306.
- D. Kaul, N. T. Nguyen and S. Venkataram, Crystal habit modifications and altered tabletting characteristics,(1992) 345-350; DOI: 10.1016/0378-5173(92)90333-W.
- H. A. Garekani, F. Sadeghi, A. Badiee, S. A. Mostafa and A. R. Rajabi-Siahboomi, Crystal habit modifications of ibuprofen and their physicochemical characteristics,(2001) 803-809; DOI: 10.1081/DDC-100107242.
- N. Rasenack and B W. Müller, Ibuprofen crystals with optimized properties,(2002) 9-24; DOI: 10.1016/S0378-5173(02)00294-6.
- K. R. Morris, U. J. Griesser, C. J. Eckhardt and J. G. Stowell, Theoretical approaches to physical transformations of active pharmaceutical ingredients during manufacturing processes,(2001) 91-114; DOI: 10.1016/S0169-409X(01)00100-4.
- Y. Kawashima and C. E. Capes, An experimental study of the kinetics of spherical agglomeration in a stirred vessel,(1974) 85-92; DOI: 10.1016/0032-5910(74)85036-9.
- Y. Kawashima, Development of spherical crystallization technique and its application to pharmaceutical systems,(1984) 145-151; DOI: 10.1007/BF02856629.
- N. Rodriguez-Hornedo, R. C. Kelly, B. D. Sinclair and J. M. Miller,(Ed. J. Swarbrick), 3rd ed., Taylor & Francis Group, New York 2006, pp. 834-857; DOI: 10.1081/E-EPT-120041347.
- A. S. Myerson and R. Ginde,, in(Ed. A. S. Myerson), 2nd ed., Butterworth-Heinemann, Woburn 2001, pp. 33-65; DOI: 10.1016/B978-075067012-8/50004-5.
- J. W. Mullin,, in(Ed. J. W. Mullin), 4th ed., Butterworth-Heinemann, Woburn 2001, pp. 216-288; DOI: 10.1016/B978-075064833-2/50008-5.
- R. F. Sekerka,, in(Eds. G. Müller, J. Métois and P. Rudolph), Elsevier, Amsterdam 2004, pp. 55-93; DOI: 10.1016/B978-044451386-1/50005-2.
- Y. Kawashima, M. Okumura and H. Takenaka, The effects of temperature on the spherical crystallization of salicylic acid,(1984) 41-47; DOI: 10.1016/0032-5910(84)85018-4.
- H. Göczo, P. Szabó-Révész, B. Farkas, M. Hasznos-Nezdei, S. F. Serwanis, A. K. Pintye-Hódi, P. Kása, Jr., I. Eros, I. Antal and S. Marto, Development of spherical crystals of acetylsalicylic acid for direct tablet-making,(2000) 1877-1881.
- A. F. Blandin, D. Mangin, A. Rivoire, J. P. Klein and J. M. Bossoutrot, Agglomeration in suspension of salicylic acid fine particles: influences of some process parameters on kinetics and agglomerate final size,(2003) 316-323; DOI: 10.1016/S0032-5910(02)00210-3.
- Y. Kawashima, K. Furukawa and H. Takenaka, The physicochemical parameters determining the size of agglomerate prepared by the wet spherical agglomeration technique,(1981) 211-216; DOI: 10.1016/0032-5910(81)80014-9.
- A. S. Bos and F. J. Zuiderweg, Kinetics of continuous agglomeration in suspension,(1985) 43-51; DOI: 10.1016/0032-5910(85)85019-1.
- Z. Sadowski, Selective spherical agglomeration of fine salt-type mineral particles in aqueous solution,(1995) 277-285; DOI: 10.1016/0927-7757(94)03042-X.
- C. Skarvelakis and G. Antonini, Kinetics of agglomerate growth in a continuous coal-oil purification process,(1995) 135-141; DOI: 10.1016/0892-6875(89)90038-1.
- B. A. Snyder and J. C. Berg, Oil-assisted agglomeration for toner deinking: Population balance model and experiments,(1997) 1480-1487; DOI: 10.1002/aic.690430611.
- J. S. Laskowski and Z. Yu, Oil agglomeration and its effect on beneficiation and filtration of low-rank/oxidized coals,(2000) 237-252; DOI: 10.1016/S0301-7516(99)90040-6.
- C. I. House and C. J. Veal, Selective recovery of chalcopyrite by spherical agglomeration,(1989) 171-184; DOI: 10.1016/0892-6875(89)90038-1.
- A. Y. Huang and J. C. Berg, Gelation of liquid bridges in spherical agglomeration,(2003) 241-252; DOI: 10.1016/S0927-7757(02)00488-0.
- S. Mahanty, J. Sruti, C. Niranjan Patra and M. E. Bhanoji Rao, Particle design of drugs by spherical crystallization techniques,(2010) 912-918.
- J. Thati and Å. C. Rasmuson, On the mechanisms of formation of spherical agglomerates,(2011) 365-379; DOI: 10.1016/j.ejps.2011.01.001.
- Y. Kawashima, F. Cui, H. Takeuchi, T. Niwa, T. Hino and K. Kiuchi, Parameters determining the agglomeration behaviour and the micromeritic properties of spherically agglomerated crystals prepared by the spherical crystallization technique with miscible solvent systems,(1995) 139-147; DOI: 10.1016/0378-5173(94)00380-N.
- J. Katta and A. C. Rasmuson, Spherical crystallization of benzoic acid,(2008) 61-69; DOI: 10.1016/j.ijpharm.2007.07.006.
- H. Zhang, Y. Chen, J. Wang and J. Gong, Investigation on the spherical crystallization process of cefotaxime sodium,(2010) 1402-1411; DOI: 10.1021/ie901001c.
- D. Amaro-González and B. Biscans, Spherical agglomeration during crystallization of an active pharmaceutical ingredient,(2002) 188-194; DOI: 10.1016/S0032-5910(02)00196-1.
- A. H. L. Chow and M. W. M. Leung, A study of the mechanisms of wet spherical agglomeration of pharmaceutical powders,(1996) 357-371; DOI: 10.3109/03639049609042001.
- M. Maghsoodi, Effect of process variables on physicomechanical properties of the agglomerates obtained by spherical crystallization technique,(2011)474-482; DOI: 10.3109/10837450.2010.492218.
- Y. Kawashima, T. Niwa, T. Handa, H. Takeuchi, T. Iwamoto and K. Itoh, Preparation of controlled-release microspheres of ibuprofen with acrylic polymers by a novel quasi-emulsion solvent diffusion method,(1989) 68-72; DOI: 10.1002/jps.2600780118.
- A. Sano, T. Kuriki, Y. Kawashima, T. Hino and T. Niwa, Particle design of tolbutamide by the spherical crystallization technique. III. Micromeritic properties and dissolution rate of tolbutamide spherical agglomerates prepared by the quasi-emulsion solvent diffusion method and the solvent change method,38 (1990) 733-739.
- K. Morishima, Y. Kawashima, H. Takeuchi, T. Niwa and T. Hino, Micromeritic characteristics and agglomeration mechanisms in the spherical crystallization of bucillamine by the spherical agglomeration and the emulsion solvent diffusion methods,(1993) 57-64; DOI: 10.1016/0032-5910(93)80041-8.
- F. Espitalier, B. Biscans and C. Laguérie, Particle design Part A: Nucleation kinetics of ketoprofen,(1997) 95-102; DOI: 10.1016/S1385-8947(97)00089-2.
- Y. Kawashima, M. Imai, H. Takeuchi, H. Yamamoto, K. Kamiya and T. Hino, Improved flowability and compactibility of spherically agglomerated crystals of ascorbic acid for direct tabletting designed by spherical crystallization process,(2003) 283-289; DOI: 10.1016/S0032-5910(02)00206-1.
- M. Nocent, L. Bertocchi, F. Espitalier, M. Baron and G. Couarraze, Definition of a solvent system for spherical crystallization of salbutamol sulfate by quasi-emulsion solvent diffusion (QESD) method,(2001) 1620-1627; DOI: 10.1002/jps.1112.
- F. Espitalier, B. Biscans and C. Laguérie, Particle design Part B: batch quasi-emulsion process and mechanism of grain formation of ketoprofen,(1997) 103-114; DOI: 10.1016/S1385-8947(97)00057-0.
- Z. Zhang, Z. Shen, J. Wang, H. X. Zhang, H. Zhao, J. F. Chen and J. Yun, Micronization of silybin by the emulsion solvent diffusion method,(2009) 116-122; DOI: 10.1016/j.ijpharm.2009.04.028.
- M. Maghsoodi and M. Esfehani, Preparation of microparticles of naproxen with Eudragit RS and Talc by spherical crystallization technique,(2009) 442-450; DOI: 10.1080/10837450902748404.
- M. Ueda, Y. Nakamura, H. Makita, Y. Imasato and Y. Kawashima, Particle design of enoxacinby spherical crystallization technique. I. Principle of ammonia diffusion system (ADS),(1990) 2537-2541.
- S. Bhadra, M. Kumar, S. Jain, S. Agrawal and G. P. Agrawal, Spherical crystallization of mefenamic acid,(2004) 66-76.
- H. G. Puechagut, J. Bianchotti and C. A. Chiale, Preparation of norfloxacin spherical agglomerates using the ammonia diffusion system,(1998) 519-523; DOI: 10.1021/js960463w.
- S. S, Kadam, K. R. Mahadik and A. R. Paradkar,, Indian Patent 183036, 14 Feb 1997.
- A. Pawar, A. Paradkar, S. Kadam and K. Mahadik, Agglomeration of ibuprofen with talc by novel crystallo-co-agglomeration technique,(2004) Article 55; DOI: 10.1208/pt050455.
- M. Maghsoodi, O. Taghizadeh, G. P. Martin and A. Nokhodchi, Particle design of naproxen-disintegrant agglomerates for direct compression by a crystallo-co-agglomeration technique,(2008) 45-54; DOI: 10.1016/j.ijpharm.2007.09.033.
- A. Pawar, A. Paradkar, S. Kadam and K. Mahadik, Crystallo-co-agglomeration: A novel technique to obtain ibuprofen-paracetamol agglomerates,(2004) Article 44; DOI: 10.1208/pt050344.
- A. Pawar, A. R. Paradkar, S. S. Kadam and K. R. Mahadik, Effect of polymers on crystallo-co-agglomeration of ibuprofen-paracetamol: Factorial design,(2007) 658-664; DOI: 10.4103/0250-474X.38471.
- P. Szabó-Révész, H. Göczo, K. Pintye-Hodi, P. Kása, Jr., I. Erõs, M. Hasznos-Nezdei and B. Farkas, Development of spherical crystal agglomerates of an aspartic acid salt for direct tablet making,(2001) 118-124; DOI: 10.1016/S0032-5910(00)00272-2.
- M. Maghsoodi, D. Hassan-Zadeh, M. Barzegar-Jalali, A. Nokhodchi and G. Martin, Improved compaction and packing properties of naproxen agglomerated crystals obtained by spherical crystallization technique,(2007) 1216-1224; DOI: 10.1080/03639040701377730.
- M. Maghsoodi and A. S. Tajalli Bakhsh, Evaluation of physico-mechanical properties of drug-excipients agglomerates obtained by crystallization,(2011) 243-249; DOI: 10.3109/10837451003610837.
- A. Nokhodchi and M. Maghsoodi, Preparation of spherical crystal agglomerates of naproxen containing disintegrant for direct tablet making by spherical crystallization technique,(2008) 54-59; DOI: 10.1208/s12249-007-9019-3.
- A. N. Usha, S. Mutalik, M. S. Reddy and A. K. Ranjith, Preparation and,, preclinical and clinical studies of aceclofenac spherical agglomerates,(2008) 674-683; DOI: 10.1016/j.ejpb.2008.06.010.
- S. Kumar, G. Chawla and A. K. Bansal, Spherical crystallization of mebendazole to improve processability,(2008) 559-568; DOI: 10.1080/10837450802310180.
- C. L. Viswanathan, S. K. Kulkarni and D. R. Kolwankar, Spherical agglomeration of mefenamic acid and nabumetone to improve micromeritics and solubility: A technical note,(2006) E122-E125, DOI: 10.1208/pt070248.
- V. R. Gupta, S. Mutalik, M. M. Patel and G. K. Jani, Spherical crystals of celecoxib to improve solubility, dissolution rate and micromeritic properties,(2007) 173-184; DOI: 10.2478/v10007-007-0014-8.
- A. R. Paradkar, A. P. Pawar, J. K. Chordiya, V. B. Patil and A. R. Ketkar, Spherical crystallization of celecoxib,(2002) 1213-1220; DOI: 10.1081/DDC-120015354.
- P. Di Martino, C. Barthélémy, F. Piva, E. Joiris, G. F. Palmieri and S. Martelli, Improved dissolution behavior of fenbufen by spherical crystallization,(1999) 1073-1081; DOI: 10.1081/DDC-100102272.
- M. Maghsoodi and F. Sadeghpoor, Preparation and evaluation of solid dispersions of piroxicam and Eudragit S100 by spherical crystallization technique,(2010) 917-925; DOI: 10.3109/03639040903585127.
- F. Cui, M. Yang, Y. Jiang, D. Cun, W. Lina, Y. Fana and Y. Kawashimab, Design of sustained-release nitrendipine microspheres having solid dispersion structure by quasi-emulsion solvent diffusion method,(2003) 375-384; DOI: 10.1016/S0168-3659(03)00275-X.
- M. Yang, F. Cui, B. You, Y. Fan, L. Wang, P. Yue and H. Yang, Preparation of sustained-release nitrendipine microspheres with Eudragit RS and Aerosil using quasi-emulsion solvent diffusion method,(2003) 103-113; DOI: 10.1016/S0378-5173(03)00209-6.
- J. Varshosaz, N. Tavakoli and F. A. Salamat, Enhanced dissolution rate of simvastatin using spherical crystallization technique,(2011) 529-535; DOI: 10.3109/10837450.2010.502175.
Language: English, Croatian, Slovenian
Page range: 1 - 14
Published on: Apr 3, 2012
Published by: Croatian Pharmaceutical Society
In partnership with: Paradigm Publishing Services
Related subjects:
© 2012 Borut Kovačič, Franc Vrečer, Odon Planinšek, published by Croatian Pharmaceutical Society
This work is licensed under the Creative Commons License.