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Effect of formulation parameters on the drug release and floating properties of gastric floating two-layer tablets with acetylsalicylic acid Cover

Effect of formulation parameters on the drug release and floating properties of gastric floating two-layer tablets with acetylsalicylic acid

Open Access
|Sep 2011

References

  1. Z. Wei, Z. Yu and D. Bi, Design and evaluation of a two-layer floating tablet for gastric retention using cisapride as a model drug, Drug Dev. Ind. Pharm. 27 (2001) 469-474; DOI: 10.1081/DDC-100104323.10.1081/DDC-100104323
  2. S. Arora, J. Ali, A. Ahuja, R. K. Khar and S. Baboota, Floating drug delivery systems: a review, AAPS PharmSciTech. 6 (2005) Article 47; DOI: 10.1208/pt060347.10.1208/pt060347
  3. Z. Rahman, M. Ali and R. K. Khar, Design and evaluation of bilayer floating tablets of captopril, Acta Pharm. 56 (2006) 49-57.
  4. R. Talukder and R. Fassihi, Gastroretentive delivery systems: a mini rewiew, Drug Dev. Ind. Pharm. 30 (2004) 1019-1028; DOI: 10.1081/DDC-200040239.10.1081/DDC-200040239
  5. S. Baumgartner, J. Kristl, F. Vrecer, P. Vodopivec and B. Zorko, Optimisation of floating matrix tablets and evaluation of their gastric residence time, Int. J. Pharm. 195 (2000) 125-135; DOI: 10.1016/SO378-5173(99)00378-6.
  6. S. Strübing, H. Metz and K. Mader, Characterization of poly(vinyl acetate) based floating matrix tablets, J. Control. Release 126 (2008) 149-155; DOI: 10.1016/j.jconrel.2007.11.013.10.1016/j.jconrel.2007.11.013
  7. G. Chawla, P. Gupta, V. Korodia and A. K. Bansal, A means to address regional variability in intestinal drug absorption, Pharm. Technol. 27 (2003) 50-68.
  8. J. Varshosaz, N. Tavakoli and F. Roozbahani, Formulation and in vitro characterization of cipro-floxacin floating and bioadhesive extended-release tablets, Drug Deliv. 13 (2006) 277-285; DOI: 10.1080/10717540500395106.10.1080/10717540500395106
  9. M. I. Tadros, Controlled-release effervescent floating matrix tablets of ciprofloxacin hydrochloride: Development, optimization and in vitro-in vivo evaluation in healthy human volunteers, Eur. J. Pharm. Biopharm. 74 (2010) 332-339; DOI: 10.1016/j.ejpb.2009.11.010.10.1016/j.ejpb.2009.11.010
  10. B. N. Singh and K. H. Kim, Floating drug delivery systems: an approach to oral controlled drug delivery via gastric retention, J. Control. Release 63 (2000) 235-259; DOI: 10.1016/S0168-3659(99)00204-7.10.1016/S0168-3659(99)00204-7
  11. N. Özdemir, Ş. Ordu and Y. Özkan, Studies of floating dosage forms of furosemide: in vitro in vivo evaluations of bilayer tablet formulations, Drug Dev. Ind. Pharm. 26 (2000) 857-866; DOI: 10.1081/DDC-100101309.10.1081/DDC-100101309
  12. United States Pharmacopeia 30/National Formulary 25, USP Convention, Rockville (MD) 2007.
  13. T. Higuchi, Mechanism of sustained-action medication: theoretical analysis of rate of release of solid drugs dispersed in solid matrices, J. Pharm. Sci. 52 (1963) 1145-1149; DOI: 10.1002/jps.2600521210.10.1002/jps.2600521210
  14. R. W. Korsmeyer, R. Gurny, E. Doelker, P. Buri and N. A. Peppas, Mechanisms of solute release from porous hydrophilic polymers, Int. J. Pharm. 15 (1983) 25-35; DOI: 10.1016/0378-5173(83)90064-9.10.1016/0378-5173(83)90064-9
  15. N. A. Peppas and J. J. Sahlin, A simple equation for the description of solute release. III: Coupling of diffusion and relaxation, Int. J. Pharm. 57 (1989) 169-172; DOI: 10.1016/0378-5173(89)90306-2.10.1016/0378-5173(89)90306-2
  16. S. Sungthongjeen, P. Sriamornsak and S. Puttipipatkhachorn, Design and evaluation of floating multi-layer coated tablets based on gas formation, Eur. J. Pharm. Biopharm. 69 (2008) 255-263; DOI: 10.1016/j.ejpb.2007.09.013.10.1016/j.ejpb.2007.09.013
  17. P. Colombo, D. Provasi, M. G. Borazza, L. Maggi and P. L. Catellani, The role of compression force in floating tablet formula optimization, Acta Pharm. Technol. 35 (1989) 168-170.
  18. P. Colombo, R. Bettini and N. A. Peppas, Observation of swelling process and diffusion front position during swelling in hydroxypropyl methylcellulose (HPMC) matrices containing a soluble drug, J. Control. Release 61 (1999) 83-91; DOI: 10.1016/S0168-3659(99)00104-2.10.1016/S0168-3659(99)00104-2
  19. N. A. Peppas, Analysis of Fickian and non-Fickian drug release from polymers, Pharm. Acta Helv. 60 (1985) 110-111.
DOI: https://doi.org/10.2478/v10007-011-0028-0 | Journal eISSN: 1846-9558 | Journal ISSN: 1330-0075
Language: English
Page range: 303 - 312
Published on: Sep 26, 2011
Published by: Croatian Pharmaceutical Society
In partnership with: Paradigm Publishing Services
Publication frequency: 4 issues per year
Related subjects:

© 2011 Canan Hasçiçek, Günseli Yüksel-Tilkan, Berna Türkmen, Nurten Özdemir, published by Croatian Pharmaceutical Society
This work is licensed under the Creative Commons License.

Volume 61 (2011): Issue 3 (September 2011)