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Design, synthesis, hydrolysis kinetics and phamacodynamic profiles of histidine and alanine conjugates of aceclofenac Cover

Design, synthesis, hydrolysis kinetics and phamacodynamic profiles of histidine and alanine conjugates of aceclofenac

By: Arun Rasheed and  C. Kumar  
Open Access
|Mar 2010

References

  1. Analgesics Anti-Inflammatory and Antipyretics, in Martindale: The Complete Drug Reference (Ed. K. Parfitt), 32nd ed., Pharmaceutical Press, London 1999, pp. 61-62.
  2. A.E. Kay and A. Alldred, Rheumatoid Arthritis and Osteoarthritis, in Clinical Pharmacy and Therapeutics (Eds. R. Walker and C. Edwards), 3rd ed., Churchill Livingstone, London 2003, pp. 791-807.
  3. A. Mishra, V. Ravichandran, P.K. Jain, V.K. Dixit and R.K. Agrawal, Synthesis, characterization and pharmacological evaluation of amide prodrugs of flubiprofen, J. Braz. Chem. Soc. 19 (2008) 89-100; DOI: 10.1590/S0103-50532008000100014.10.1590/S0103-50532008000100014
  4. A. Mishra, V. Ravichandran, P.K. Jain, V.K. Dixit and R.K. Agrawal, Synthesis, characterization and pharmacological evaluation of amide prodrugs of ketorolac, Eur. J. Med. Chem. 43 (2008) 2464-2472; DOI: 10.1016/j.ejmech.2007.09.011.10.1016/j.ejmech.2007.09.011
  5. D. Bhosle, S. Bharambe, N. Gairola and S.S. Dhaneshwar, Mutual prodrug concept: fundamentals and applications, Indian J. Pharm. Sci. 68 (2006) 286-294; DOI: 10.4103/0250-474X.26654.10.4103/0250-474X.26654
  6. A. Rasheed and C.K.A. Kumar, Novel approaches on prodrug based drug design, Pharm. Chem. J. 42 (2008) 677-686; DOI: 10.1007/s11094-009-0213-3.10.1007/s11094-009-0213-3
  7. S.D. Roy and E. Manoukian, Permeability of ketorolac acid and its ester analogs (prodrug) through human cadaver skin, J. Pharm. Sci. 83 (1994) 1548-1553; DOI: 10.1002/jps.2600831106.10.1002/jps.2600831106
  8. J.R. Idle, P. Millburn and R.T. Williams, Taurine conjugates as metabolites of arylacetic acids in the ferret, Xenobiotica 8 (1978) 253-264; DOI: 10.3109/00498257809056147.10.3109/00498257809056147
  9. N. Gairola, D. Nagpal, S.S. Dhaneshwar, S.R. Dhaneshwar and S.C. Chaturvedi, Synthesis, hydrolysis kinetics and pharmacodynamic profiles of novel prodrugs of flubiprofen, Indian J. Pharm. Sci. 67 (2005) 369-373.
  10. A. Rasheed, V. Ravichandran and D.V. Kohli, Ampicillin prodrugs: amide conjugates from amino acids, peptide and ampicillin, Pharmazie 54 (1999) 857-858.
  11. N.W. Nielsenw and H. Bundgaard, Glycolamide esters as biolabile prodrugs of carboxylic acid agents: synthesis, stability, bioconversion, and physicochemical properties, J. Pharm. Sci. 77 (1988) 285-298; DOI: 10.1002/jps.2600770402.10.1002/jps.2600770402
  12. C.A. Winter, E.A. Risely and G.W. Nuss, Carregeenan induced oedema in hind paw of the rat as assay for anti-inflammatory drugs, Exp. Biol. Med. 111 (1962) 544-547.10.3181/00379727-111-27849
  13. S.K. Kulkarni, Heat and other physiological stress-induced analgesia: catecholamine mediated and naloxone reversible response, Life Sci. 27 (1980) 185-188; DOI: 10.1016/0024-3205(80)90136-8.10.1016/0024-3205(80)90136-8
  14. R.K. Goyal, A. Chakrabarti and A.K. Sanyal, The effect of biological variables on the anti-ulcerogenic effect of vegetable plantain banana, Planta Med. 29 (1985) 85-88; DOI: 10.1055/s-2007-969412.10.1055/s-2007-9694124034739
  15. M. Yagmurca, M. Ucar, E. Fadillioglu, H. Erdogan and F. Ozturk, The effects of nitric oxide on rat stomach injury induced by acetylsalicylic acid, Turk. J. Med. Sci. 39 (2009) 13-19; DOI: 10.3906/sag-0712-22.10.3906/sag-0712-22
DOI: https://doi.org/10.2478/v10007-010-0003-1 | Journal eISSN: 1846-9558 | Journal ISSN: 1330-0075
Language: English
Page range: 99 - 109
Published on: Mar 13, 2010
Published by: Croatian Pharmaceutical Society
In partnership with: Paradigm Publishing Services
Publication frequency: 4 issues per year
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© 2010 Arun Rasheed, C. Kumar, published by Croatian Pharmaceutical Society
This work is licensed under the Creative Commons License.

Volume 60 (2010): Issue 1 (March 2010)