Synthesis and evaluation of anti-inflammatory, analgesic, ulcerogenic and lipid peroxidation properties of ibuprofen derivatives
By: Mohammad Amir and Shikha Kumar
Open Access
|Feb 2007References
- M. B. Kimmey, NSAID, ulcers and prostaglandins,19 (1992) 68-73.
- C. J. Smith, Y. Zhang, C. M. Koboldt, J. Muhammad, B. S. Zwefel, A. Shaffer, J. J. Talley, J. L. Masferrer, K. Serbert and P. C. Isakson, Pharmacological analysis of cyclo-oxygenase-1 in in-flammation,95 (1998) 13313-13318.
- C. Hawkey, L. Laine, T. Simon, A. Beaulieu, J. Maldonado-Cocco, E. Acevedo, A. Shahane, H. Quan, J. Bolognese and E. Mortensen, Comparison of the effect of rofecoxib, ibuprofen and placebo on the gastroduodenal mucosa of patients with osteoarthritis: A randomized, double blind, placebo-controlled trial,43 (2000) 370-377.
- T. D. Warner, F. Giuliano, I. Vaynovie, A. Bukasa, J. A. Mitchell and J. R. Vave, Non-steroid drug selectivities for cyclo-oxygenase-1 rather than cyclo-oxygenase-2 are associated with human gastro-intestinal toxicity: A fullanalysis,96 (1999) 7563-7568.
- F. L. Lanza, A guideline for the treatment and prevention of NSAID-induced ulcers,93 (1998) 2037-2046.
- A. S. Kalgutkar, A. B. Marnett, B. C. Crews, R. P. Remmel and L. J. Marnett, Ester and amide derivatives of the nonsteroidal antiinflammatory drug, indomethacin, as selective cyclo-oxygenase-2 inhibitor,43 (2000) 2860-2870.
- M. Duflos, M. R. Nourrisson, J. Brelet, J. Courant, G. Le Baut, N. Grimaud and J. Y. Petit, N-Pyridinyl-indole-3-(alkyl) carboxamides and derivatives as potential systemic and topical inflammation inhibitors,36 (2001) 545-553.
- M. Amir and S. Kumar, Anti-inflammatory and gastro sparing activity of some new indomethacin derivatives,338 (2005) 24-31.
- F. A. Omar, N. M. Mahfouz and M. A. Rahman, Design, synthesis and anti-inflammatory activity of some 1,3,4-oxadiazole derivatives,31 (1996) 819-825.
- M. Amir, A. Oberoi and S. Alam, Synthesis and anti-inflammatory activity of some new 6-methoxy-β-methyl-2-naphthalene acetic acid derivatives,38B (1999) 237-239.
- E. Palaska, G. Sahin, P. Kelicen, N. T. Durlu and G. Altinok, Synthesis and anti-inflammatory activity of 1-acylthiosemicarbazide: 1,3,4-oxadiazoles, 1,3,4-thiadiazoles and 1,2,4-triazole-3-thiones,57 (2002) 101-107.
- B. Furniss, A. H. Hannaford, P. W. G. Smith and A. R. Tatchell,, 5th ed., Addison Wesley Longman, New Delhi (1998 pp. 1077.
- C. A. Winter, E. A. Risley and G. N. Nuss, Carrageenin-induced edema in hind paw of the rat as an assay for anti-inflammatory drugs,111 (1962) 544-547.
- A. Kumar, D. Bansal, K. Bajaj, S. Sharma, Archana and V. K. Srivastava, Synthesis of some newer derivatives of 2-amino benzoic acid as potent anti-inflammatory and analgesic agents,11 (2003) 5281-5291.
- V. Cioli, S. Putzolu, V. Rossi, P. Sorza Barcellona and C. Corradino, The role of direct tissue contact in the production of gastro-intestinal ulcers by anti-inflammatory drugs in rats,50 (1979) 283-289.
- H. Ohkawa, N. Ohishi and K. Yagi, Assay for lipid peroxides in animal tissues by thiobarbituric acid reaction,95 (1979) 351-358.
- B. Galunska, K. Marazova, T. Yankova, A. Popov, P. Frangov, I. Krushkov and D. I. Massa, Effect of paracetamol and propacetamol on gastric mucosal damage and gastric lipid per oxidation caused by acetylsalicylic acid in rats,46 (2002) 141-148.
- Y. Naito, T. Yoshikawa, N. Yoshida and M. Kondo, Role of oxygen radical and lipid peroxidation in indomethacin-induced gastric mucosal injury,43 (Suppl. 9) (1998) 30S-34S.
- T. Pohle, T. Brzozowski, J. C. Becker, I. R. Vander Voort, A. Markmann, S. J. Konturek, A. Moniczewski, W. Domschke and J. W. Konturek, Role of reactive oxygen metabolites in aspirin-induced gastric damage in humans, gastroprotection by vitamin,15 (2001) 677-687.
Language: English
Page range: 31 - 45
Published on: Feb 28, 2007
Published by: Croatian Pharmaceutical Society
In partnership with: Paradigm Publishing Services
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© 2007 Mohammad Amir, Shikha Kumar, published by Croatian Pharmaceutical Society
This work is licensed under the Creative Commons License.