Have a personal or library account? Click to login
Preparation and in vivo evaluation of a gel-based nasal delivery system for risperidone Cover

Preparation and in vivo evaluation of a gel-based nasal delivery system for risperidone

Open Access
|Oct 2016

References

  1. 1. T. Cabaleiro, D. Ochoa, R. López-Rodríguez, M. Román, J. Novalbos, C. Ayuso and F. Abad-Santos, Effect of polymorphisms on the pharmacokinetics, pharmacodynamics, and safety of risperidone in healthy volunteers, Hum. Psychopharmacol. 29 (2014) 459-469; DOI: 10.1002/hup.2420.10.1002/hup.242025042870
  2. 2. J. L. Sun, Q. X. Chen, S. Tian, F. R. Meng, Y. Lv and G. H. Du, Absorption of risperidone polymorphs administrated orally in rats, Chin. Pharm. J. 46 (2011) 1919-1922.
  3. 3. T. K. Vyas, A. Shahiwala, S. Marathe and A. Misra, Intranasal drug delivery for brain targeting, Curr. Drug Deliv. 2 (2005) 165-175; DOI: 10.2174/1567201053586047.10.2174/156720105358604716305417
  4. 4. C. R. Behl, H. K. Pimplaskar, A. P. Sileno, J. deMeireles and V. D. Romeo, Effects of physicochemical properties and other factors on systemic nasal drug delivery, Adv. Drug Deliv. Rev. 29 (1998) 89-116; DOI: doi:10.1016/S0169-409X(97)00063-X.
  5. 5. M. Kumar, A. Misra, A. K. Babbar, A. K. Mishra, P. Mishra and K. Pathak, Intranasal nanoemulsion based brain targeting drug delivery system of risperidone, Int. J. Pharm. 358 (2008) 285-291; DOI: 10.1016/j.ijpharm.2008.03.029.10.1016/j.ijpharm.2008.03.02918455333
  6. 6. W. N. Ma and F. G. Gu, Effect of pH on the chemical stability, solubility and oil-water partition coefficient of risperidone, Centr. South Pharm. 13 (2015) 473-476; DOI: 10.7539/j.issn.1672-2981.2015.05.006.
  7. 7. H. S. Mahajan, S. K. Shah and S. J. Surana, Nasal in situ gel containing hydroxy propyl β-cyclodextrin inclusion complex of arthemeter: development and in vitro evaluation, J. Incl. Phenom. Macrocycl. Chem. 70 (2011) 49-58; DOI: 10.1007/s10847-010-9861-x.10.1007/s10847-010-9861-x
  8. 8. C. Tas, C. K. Ozkan, A. Savaser, Y. Ozkan, U. Tasdemir and H. Altunay, Nasal absorption of metoclopramide from different Carbopol 981 based formulations: In vitro, ex vivo and in vivo evaluation, Eur. J. Pharm. Biopharm. 64 (2006) 246-254; DOI: 10.1016/j.ejpb.2006.05.017.10.1016/j.ejpb.2006.05.01716870409
  9. 9. F. G. Gu, F. D. Cui and Y. L. Gao, Preparation of prostaglandin E1-hydroxypropyl-β-cyclodextrin complex and its nasal delivery in rats, Int. J. Pharm. 290 (2005) 101-108; DOI: 10.1016/j. ijpharm.2004.11.021.
  10. 10. X. G. Jiang, J. B. Cui, X. L. Fang, Y. Wei and N. Z. Xi, Toxicity of drugs on nasal mucocilia and the method of its evaluation, Acta. Pharm. Sin. 30 (1995) 848-853; DOI: 10.3321/j.issn:0513-4870.1995.11.009.
  11. 11. M. Jug, I. Kos and M. Bećirević-Laćan, The pH-dependent complexation between risperidone and hydroxypropyl-β-cyclodextrin, J. Incl. Phenom. Macrocycl. Chem. 64 (2009) 163-171; DOI: 10.1007/ s10847-009-9549-2.10.1007/s10847-009-9549-2
  12. 12. T. Yang, A. Hussain, J. Paulson, T. J. Abbruscato and F. Ahsan, Cyclodextrinsin nasal delivery of low molecular weight heparins: in vivo and in vitro studies, Pharm. Res. 21 (2004) 1127-1136; DOI: 10.1023/B:PHAM.0000032998.84488.7a.10.1023/B:PHAM.0000032998.84488.7a
  13. 13. E. Marttin, J. C. Vethoef and F. W. H. M. Merkus, Efficacy safety and mechanism of cyclodextrins as absorption enhancers in nasal delivery of peptide and protein drugs, J. Drug Targeting 6 (1998) 17-36; DOI: 10.3109/10611869808997878.10.3109/106118698089978789769018
  14. 14. G. Rathnam, N. Narayanan and R. Ilavarasan, Carbopol-based gels for nasal delivery of progesterone, AAPS Pharm. Sci. Tech. 9 (2008) 1078-1082; DOI: 10.1208/s12249-008-9144-7.10.1208/s12249-008-9144-7262826518850277
  15. 15. F. G.. Gu, D. Hao, G. D. L. Meng, C. Z. Wu and Y. Wang, Preparation of bisoprolol fumarate nasal spray and its nasal delivery in rats, Pak. J. Pharm. Sci. 28 (2015) 2173-2178.
DOI: https://doi.org/10.1515/acph-2016-0047 | Journal eISSN: 1846-9558 | Journal ISSN: 1330-0075
Language: English
Page range: 555 - 562
Accepted on: Aug 3, 2016
Published on: Oct 15, 2016
Published by: Croatian Pharmaceutical Society
In partnership with: Paradigm Publishing Services
Publication frequency: 4 issues per year
Related subjects:

© 2016 Fugen Gu, Weina Ma, Gendalai Meng, Chunzhi Wu, Yi Wang, published by Croatian Pharmaceutical Society
This work is licensed under the Creative Commons Attribution-NonCommercial-NoDerivatives 4.0 License.